Matched molecular pairs as a medicinal chemistry tool: miniperspective E Griffen, AG Leach, GR Robb, DJ Warner Journal of medicinal chemistry 54 (22), 7739-7750, 2011 | 282 | 2011 |
Molecular basis of peripheral vs central benzodiazepine receptor selectivity in a new class of peripheral benzodiazepine receptor ligands related to alpidem M Anzini, A Cappelli, S Vomero, G Giorgi, T Langer, G Bruni, MR Romeo, ... Journal of medicinal chemistry 39 (21), 4275-4284, 1996 | 117 | 1996 |
Novel, potent, and selective 5-HT3 receptor antagonists based on the arylpiperazine skeleton: synthesis, structure, biological activity, and comparative molecular field … M Anzini, A Cappelli, S Vomero, G Giorgi, T Langer, M Hamon, N Merahi, ... Journal of medicinal chemistry 38 (14), 2692-2704, 1995 | 103 | 1995 |
Design, Synthesis, Structural Studies, Biological Evaluation, and Computational Simulations of Novel Potent AT1 Angiotensin II Receptor Antagonists Based on the … A Cappelli, G Pericot Mohr, A Gallelli, M Rizzo, M Anzini, S Vomero, ... Journal of medicinal chemistry 47 (10), 2574-2586, 2004 | 102 | 2004 |
Novel potent and selective central 5-HT3 receptor ligands provided with different intrinsic efficacy. 1. Mapping the central 5-HT3 receptor binding site by arylpiperazine … A Cappelli, M Anzini, S Vomero, L Mennuni, F Makovec, E Doucet, ... Journal of medicinal chemistry 41 (5), 728-741, 1998 | 97 | 1998 |
Further studies on imidazo [4, 5-b] pyridine AT1 angiotensin II receptor antagonists. Effects of the transformation of the 4-phenylquinoline backbone into 4 … A Cappelli, G Pericot Mohr, G Giuliani, S Galeazzi, M Anzini, L Mennuni, ... Journal of medicinal chemistry 49 (22), 6451-6464, 2006 | 90 | 2006 |
Mapping and fitting the peripheral benzodiazepine receptor binding site by carboxamide derivatives. Comparison of different approaches to quantitative ligand− receptor … M Anzini, A Cappelli, S Vomero, M Seeber, MC Menziani, T Langer, ... Journal of medicinal chemistry 44 (8), 1134-1150, 2001 | 88 | 2001 |
Novel and highly potent 5-HT3 receptor agonists based on a pyrroloquinoxaline structure G Campiani, A Cappelli, V Nacci, M Anzini, S Vomero, M Hamon, ... Journal of medicinal chemistry 40 (22), 3670-3678, 1997 | 87 | 1997 |
Synthesis and biological evaluation of amidine, guanidine, and thiourea derivatives of 2-amino (6-trifluoromethoxy) benzothiazole as neuroprotective agents potentially useful … M Anzini, A Chelini, A Mancini, A Cappelli, M Frosini, L Ricci, M Valoti, ... Journal of medicinal chemistry 53 (2), 734-744, 2010 | 80 | 2010 |
Synthesis and characterization of a new benzofulvene polymer showing a thermoreversible polymerization behavior A Cappelli, G Pericot Mohr, M Anzini, S Vomero, A Donati, M Casolaro, ... The Journal of Organic Chemistry 68 (24), 9473-9476, 2003 | 76 | 2003 |
Design, Synthesis, and Biological Evaluation of AT1 Angiotensin II Receptor Antagonists Based on the Pyrazolo[3,4-b]pyridine and Related Heteroaromatic … A Cappelli, C Nannicini, A Gallelli, G Giuliani, S Valenti, GP Mohr, ... Journal of medicinal chemistry 51 (7), 2137-2146, 2008 | 71 | 2008 |
Further studies on the interaction of the 5-hydroxytryptamine3 (5-HT3) receptor with arylpiperazine ligands. Development of a new 5-HT3 receptor ligand showing potent … A Cappelli, A Gallelli, M Manini, M Anzini, L Mennuni, F Makovec, ... Journal of medicinal chemistry 48 (10), 3564-3575, 2005 | 70 | 2005 |
Aromatase and 5-alpha reductase gene expression: modulation by pain and morphine treatment in male rats AM Aloisi, I Ceccarelli, P Fiorenzani, M Maddalena, A Rossi, V Tomei, ... Molecular Pain 6, 1744-8069-6-69, 2010 | 66 | 2010 |
Labeling and Evaluation of N-[11C]Methylated Quinoline-2-carboxamides as Potential Radioligands for Visualization of Peripheral Benzodiazepine Receptors M Matarrese, RM Moresco, A Cappelli, M Anzini, S Vomero, P Simonelli, ... Journal of medicinal chemistry 44 (4), 579-585, 2001 | 66 | 2001 |
Structural manipulation of benzofulvene derivatives showing spontaneous thermoreversible polymerization. Role of the substituents in the modulation of polymer properties A Cappelli, S Galeazzi, G Giuliani, M Anzini, A Donati, L Zetta, R Mendichi, ... Macromolecules 40 (9), 3005-3014, 2007 | 63 | 2007 |
Mapping the peripheral benzodiazepine receptor binding site by conformationally restrained derivatives of 1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)-3 … A Cappelli, M Anzini, S Vomero, PG De Benedetti, MC Menziani, G Giorgi, ... Journal of medicinal chemistry 40 (18), 2910-2921, 1997 | 63 | 1997 |
1, 5-Diarylpyrrole-3-acetic acids and esters as novel classes of potent and highly selective cyclooxygenase-2 inhibitors M Biava, GC Porretta, A Cappelli, S Vomero, F Manetti, M Botta, ... Journal of medicinal chemistry 48 (9), 3428-3432, 2005 | 62 | 2005 |
Cyclooxygenase-2 inhibitors. 1, 5-diarylpyrrol-3-acetic esters with enhanced inhibitory activity toward cyclooxygenase-2 and improved cyclooxygenase-2/cyclooxygenase-1 selectivity M Biava, GC Porretta, G Poce, S Supino, S Forli, M Rovini, A Cappelli, ... Journal of medicinal chemistry 50 (22), 5403-5411, 2007 | 57 | 2007 |
Synthesis, biological evaluation, and enzyme docking simulations of 1, 5-diarylpyrrole-3-alkoxyethyl ethers as selective cyclooxygenase-2 inhibitors endowed with anti … M Anzini, M Rovini, A Cappelli, S Vomero, F Manetti, M Botta, L Sautebin, ... Journal of medicinal chemistry 51 (15), 4476-4481, 2008 | 56 | 2008 |
Design, synthesis, and structure–affinity relationship studies in NK1 receptor ligands based on azole-fused quinolinecarboxamide moieties A Cappelli, G Giuliani, M Anzini, D Riitano, G Giorgi, S Vomero Bioorganic & medicinal chemistry 16 (14), 6850-6859, 2008 | 55 | 2008 |